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Mendeleev Communications, 2020, Volume 30, Issue 3, Pages 347–349
DOI: https://doi.org/10.1016/j.mencom.2020.05.029 (Mi mendc1193) 		 
This article is cited in 8 scientific papers (total in 8 papers)

Communications

Synthesis of new physiologically active (2-oxoimidazolidin-5-yl)indoles

L. A. Sviridovaa, P. S. Protopopovab, M. G. Akimovc, M. S. Dudinac, E. K. Melnikovaab, K. A. Kochetkovbd

a Department of Chemistry, M.V. Lomonosov Moscow State University, Moscow, Russian Federation
b A.N. Nesmeyanov Institute of Organoelement Compounds of Russian Academy of Sciences, Moscow, Russian Federation
c M.M. Shemyakin–Yu.A. Ovchinnikov Institute of Bioorganic Chemistry, Russian Academy of Sciences, Moscow, Russian Federation
d D.Mendeleev University of Chemical Technology of Russia, Moscow, Russian Federation
Full-text PDF (288 kB) Citations (8)
DOI: https://doi.org/10.1016/j.mencom.2020.05.029
Abstract: Boron trifluoride-catalyzed amidoalkylation of indole derivatives with 5-hydroxy-1-phenylimidozolidin-2-one affords new biheterocycles with a direct C–C bond. Among them, 3- or 2-(2-oxoimidazolidin-5-yl)indoles manifest antiinflammatory activity with relatively low toxicity.
Keywords: amidoalkylation, biheterocycles, 3- or 2-(2-oxoimidazolidin-5-yl)indoles, anti-inflammatory activity, indoles, imidazolylindoles.
Document Type: Article
Language: English
Supplementary materials:
Supplementary_data_1.pdf (1.4 Mb)


Citation: L. A. Sviridova, P. S. Protopopova, M. G. Akimov, M. S. Dudina, E. K. Melnikova, K. A. Kochetkov, “Synthesis of new physiologically active (2-oxoimidazolidin-5-yl)indoles”, Mendeleev Commun., 30:3 (2020), 347–349
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  • https://www.mathnet.ru/eng/mendc1193
  • https://www.mathnet.ru/eng/mendc/v30/i3/p347
    • This publication is cited in the following 8 articles:
    1. Yao Cheng, Tsz Tin Yu, Mohan Bhadbhade, David StC. Black, Naresh Kumar, “Synthesis of Indoles through C2–C3 Bond Formation Using Lawesson's Reagent”, J. Org. Chem., 2025  crossref
    2. NIKHIL KHANDALE, MANGESH S. GHODKE, “EXPLORING POTENTIAL OF INDOLE DERIVATIVES: A BRIEF REVIEW”, Int J Pharm Pharm Sci, 2023, 1  crossref
    3. Konstantin A. Kochetkov, Olga N. Gorunova, Natalia A. Bystrova, “Biologically Oriented Hybrids of Indole and Hydantoin Derivatives”, Molecules, 28:2 (2023), 602  crossref
    4. K. A. Kochetkov, O. N. Gorunova, N. A. Bystrova, “5-Hydroxy-1-phenylimidazolidine-2-thione as a new amidoalkylating agent for heterocyclic compounds”, Russ Chem Bull, 71:3 (2022), 587  crossref
    5. Grigorii K. Sterligov, Alexandra A. Ageshina, Sergey A. Rzhevskiy, Olga V. Shurupova, Maxim A. Topchiy, Lidiya I. Minaeva, Andrey F. Asachenko, “One-Pot Modified Madelung Synthesis of 3-Tosyl- and 3-Cyano-1,2-disubstituted Indoles”, ACS Omega, 7:43 (2022), 38505  crossref
    6. K. A. Kochetkov, O. N. Gorunova, N. A. Bystrova, P. V. Dudina, M. G. Akimov, “Synthesis and physiological activity of new imidazolidin-2-one bis-heterocyclic derivatives”, Russ Chem Bull, 71:11 (2022), 2395  crossref
    7. Almir S. Gazizov, Andrey V. Smolobochkin, Elizaveta A. Kuznetsova, Dinara S. Abdullaeva, Alexander R. Burilov, Michail A. Pudovik, Alexandra D. Voloshina, Victor V. Syakaev, Anna P. Lyubina, Syumbelya K. Amerhanova, Julia K. Voronina, “The Highly Regioselective Synthesis of Novel Imidazolidin-2-Ones via the Intramolecular Cyclization/Electrophilic Substitution of Urea Derivatives and the Evaluation of Their Anticancer Activity”, Molecules, 26:15 (2021), 4432  crossref
    8. G. A. Chesnokov, A. A. Ageshina, A. V. Maryanova, S. A. Rzhevskiy, P. S. Gribanov, M. A. Topchiy, M. S. Nechaev, A. F. Asachenko, “Nitromethane as a reagent for the synthesis of 3-nitroindoles from 2-haloarylamine derivatives”, Russ Chem Bull, 69:12 (2020), 2370  crossref
    Citing articles in Google Scholar: Russian citations, English citations
    Related articles in Google Scholar: Russian articles, English articles
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