Abstract:
Starting from 1,3-dinitro-5-trifluoromethylbenzene, a pioneering synthesis and dimethylaminomethylation of new 2-aryl-4-hydroxy-6-trifluoromethylindoles have been performed. The study of fungicidal activity has revealed the effect of dimethylaminomethyl group position on fungitoxic properties.
Citation:
M. D. Dutov, V. V. Kachala, B. I. Ugrak, V. A. Korolev, S. V. Popkov, D. R. Aleksanyan, O. N. Rusina, K. G. Aleksanyan, V. N. Koshelev, “Synthesis and fungicidal activity of new 4-hydroxy-6-trifluoromethyl-2-phenylindoles”, Mendeleev Commun., 28:4 (2018), 437–438
Linking options:
https://www.mathnet.ru/eng/mendc1793
https://www.mathnet.ru/eng/mendc/v28/i4/p437
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G. A. Chesnokov, A. A. Ageshina, A. V. Maryanova, S. A. Rzhevskiy, P. S. Gribanov, M. A. Topchiy, M. S. Nechaev, A. F. Asachenko, “Nitromethane as a reagent for the synthesis of 3-nitroindoles from 2-haloarylamine derivatives”, Russ Chem Bull, 69:12 (2020), 2370
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L. A. Sviridova, P. S. Protopopova, M. G. Akimov, M. S. Dudina, E. K. Melnikova, K. A. Kochetkov, “Synthesis of new physiologically active (2-oxoimidazolidin-5-yl)indoles”, Mendeleev Commun., 30:3 (2020), 347–349
D. V. Belyaev, D. L. Chizhov, M. I. Kodess, M. A. Ezhikova, G. L. Rusinov, V. N. Charushin, “Synthesis of 2-(polyfluoromethyl)pyrimido-[1,2-a]benzimidazole-4-carbaldehyde derivatives”, Mendeleev Commun., 29:3 (2019), 249–251