X. He, J. Sui, J. Xu, Z. Wang, T. Yuan, D. Liu, L. Wang, Q. Zhu, “Mild cuprous halide mediated direct C3 monohalogenation of indoles”, Mendeleev Commun., 35:2 (2025), 214

Loading [MathJax]/jax/output/SVG/config.js

Mendeleev Communications

RUS ENG

JOURNALS PEOPLE ORGANISATIONS CONFERENCES SEMINARS VIDEO LIBRARY PACKAGE AMSBIB

JavaScript is disabled in your browser. Please switch it on to enable full functionality of the website

	General information
	Latest issue
	Archive

	Search papers
	Search references

	RSS
	Latest issue
	Current issues
	Archive issues
	What is RSS

Mendeleev Commun.:
Year:
Volume:
Issue:
Page:
	Find

Personal entry:
Login:
Password:
	Save password
	Enter
	Forgotten password?
	Register

Mendeleev Communications, 2025, Volume 35, Issue 2, Pages 214–216
DOI: https://doi.org/10.71267/mencom.7609 (Mi mendc1359)

Communications

Mild cuprous halide mediated direct C³ monohalogenation of indoles

X. He^a, J. Sui^b, J. Xu^a, Z. Wang^a, T. Yuan^a, D. Liu^a, L. Wang^a, Q. Zhu^c

^a School of Chemical and Pharmaceutical Engineering, Changzhou Vocational Institute of Engineering, 213164 Changzhou, P.R. China
^b Nanjing Customs Testing Center for Dangerous Goods and Packaging, 213100 Changzhou, China
^c Department of Medicinal Chemistry, China Pharmaceutical University, 210009 Nanjing, China

Full-text PDF (295 kB)

References:

PDF

HTML

DOI: https://doi.org/10.71267/mencom.7609

Graphic abstract: Mild cuprous halide mediated direct C<sup>3</sup> monohalogenation of indoles

Abstract: Treatment of indoles with cuprous halide–N-fluorobenzenesulfonimide system in MeCN at room temperature affords the corresponding C³-halogenated derivatives. Cuprous halide acts as a dual-function reagent serving both as the halogen source and the promoter.

Keywords: indole derivatives, halogenation, cuprous halide, N-fluorobenzenesulfonimide, mild conditions.

Received: 02.09.2024
Accepted: 16.10.2024

Document Type: Article

Language: English

*Supplementary materials:*
		Supplementary_data_1.pdf	(5.1 Mb)

Citation: X. He, J. Sui, J. Xu, Z. Wang, T. Yuan, D. Liu, L. Wang, Q. Zhu, “Mild cuprous halide mediated direct C³ monohalogenation of indoles”, Mendeleev Commun., 35:2 (2025), 214–216

Linking options:

https://www.mathnet.ru/eng/mendc1359

https://www.mathnet.ru/eng/mendc/v35/i2/p214

Citing articles in Google Scholar: Russian citations, English citations
Related articles in Google Scholar: Russian articles, English articles

Statistics & downloads:
Abstract page:	75
Full-text PDF :	4
References:	13

Что такое QR-код?

Registration to the website

Logotypes